Диссертация (Синтез, свойства, структура и биологическая активность новых S и N производных пиримидина), страница 56
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Chattopadhyay, K.Ray // Tetrahedron Lett. – 2008. – Vol. 49. – P. 4405-4408.277. Regiospecific addition of uracil to acrylates catalyzed by alkaline protease fromBacillus subtilis / Y. Cai, J.Y. Wu, N. Wang [et al.] // Chin. Chem. Lett. – 2004. –Vol. 15. – P. 594-596.278. Scaffold hopping: exploration of acetanilide-containing uracil analogues as potential NNRTls / D.A. Babkov, V.T. Valuev-Elliston, M.P. Paramonova [et al.] //Bioorg. Med. Chem. – 2015.
– Vol. 23. – P. 1069-1081.279. Semenov, V.E. Synthesis of acyclic and macrocyclic analogs of di-, tri-, andtetranucleotides / V.E. Semenov, V.D. Akamsin, V.S. Reznik // Rus. J. Gen.Chem. – 2007. – Vol. 77. – P. 1430-1440.280. Seth, A. Topical liposomal gel of idoxuridine for the treatment of herpes simplex: pharmaceutical and clinical implications / A. Seth, A. Misra, D. Umrigar //Pharm.
Dev. Technol. – 2004. – Vol. 9. – P. 277-289.281. Singh, P. A practical approach for spiro- and 5-monoalkylated barbituric acids /381P. Singh, K. Paul // J. Heterocyclic Chem. – 2006. – Vol. 43. – P. 607-612.282. Sosnowski, М. A comparison of microware-accelerated and conventionallyheated iodination reactions of some arenes and heteroarenes, using ortho-periodicacid as the oxidant / М. Sosnowski, L. Skulski // Molecules.
- 2005. - Vol. 2. - P.401-406.283. Stereoselective synthesis of new bicyclic N,O-iso-homonucleoside analogues /B. Richichi, S. Cicchi, U. Chiacchio [et al.] // Tetrahedron. – 2003. – Vol. 59. – P.5231-5240.284. Structure-activity relationship studies on N3-substituted willardiine derivativesacting as AMPA or kainate receptor antagonists / N.P.
Dolman, J.C.A. More, A.Alt [et al.] // J. Med. Chem. – 2006. – Vol. 49. – P. 2579-2592.285. Structure and structure-acrivity relationships of 1-arylmethyl-5-aryl-6methyluracils as potent gonadotropin-releasing hormone receptor antagonists /Zh. Guo, Y.-F. Zhu, T.D. Gross [et al.] // J. Med. Chem. – 2004. – Vol. 47. – P.1259-1271.286. Subclinical coronary atherosclerosis predicts cardiovascular risk in differentstages of hypertension: result of the heinz nixdorf recall study / R. Erbel, N.
Lehmann, S. Möhlenkamp [et al.] // Hypertension. – 2012. – Vol. 59. – P. 44–53.287. Substituted benzyl-pyrimidines targeting thymidine monophosphate kinase ofMycobacterium tuberculosis: synthesis aand in vitro anti-mycobacterial activity /C. Gasse, D. Douguet, V. Huteau [et al.] // Bioorg. Med. Chem. – 2008. – Vol. 16.– P.
6075-6085.288. 7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists ofthe transirnt receptor potential ankyrin 1 (TRPA1) channel: a promising approachfor treating pain and inflammation / P.G. Baraldi, R. Romagnoli, G.
Saponaro [etal.] // Bioorg. Med. Chem. – 2012. – Vol. 20. - P. 1690-1698.289. Switching between reaction pathways by an alcohol cosolvent effect: SmI2ethylene glycol vs SmI2-H2O mediated synthesis of uracils / M. Szostak, M.Spain, B. Sautier, D.J. Procter // Org. Lett. – 2014. – Vol. 16. – P. 5694-5697.290.
Synthesis aerobic cytotoxity, and radiosensitizing activity of novel 2,4-382dinitrophenylamine tethered 5-fluorouracil and hydroxyurea / A. Khalaj, A.R.Doroudi, S.N. Ostad [et al.] // Bioorg. Med. Chem. Lett. – 2006. – Vol. 16. – P.6034-6038.291. Synthesis and anti-HCMV activity of 1-[ω-(phenoxy)alkyl]uracil derivativesand analogues thereof / M. S. Novikov, D. A. Babkov, M.
P. Paramonova [et al.]// Bioorg. Med. Chem. – 2013. – Vol. 21. – P. 4151-4157.292. Synthesis and anti-HIV-1 evaluation of new Sonogashira-modified Emivirine(MKC-442) analogues / K. Danel, P.T. Jorgensen, E.B. Pedersen [et al.] // Helvetica Chimica Acta. – 2009. – Vol. 92. - P. 1385-1403.293. Synthesis and antimicrobial activity of some novel 5-alkyl-6-substituted uracilsand related derivatives / A.A. Al-Turkistani, O.A. Al-Deeb, N.R. El-Brollosy,A.A. El-Emam // Molecules.
– 2011. – Vol. 16. – P. 4764-4774.294. Synthesis & antimicrobial activity of some novel pyrimidine-2,4(1H,3H)diones / O. Sharma, B. Shrivastava, R.K. Singla, V. Bhat G // Indo-Global J.Pharm. Sciences. – 2011. – Vol. 1. – P. 252-257.295.Synthesisandantiviralactivityofdeoxyanalogsof1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thimine (HEPT) as potent and selective anti-HIV-1 agents / H. Tanaka, H. Takashima, M. Ubasawa [et al.] // J. Med. Chem.– 1992. – Vol. 35. – P.
4713-4719.296. Synthesis and antiviral activity of 4H-[1,2,5]oxadiazolo[3,4-d]pyrimidine-5,7dione 1-oxide nucleosides / J.O. Shi, J. Gao, Y.P. Wang, Q.Z. Yao // ChineseChemical Lett. – 2009. – Vol. 20. - P. 404-406.297. Synthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors / R. Edupuganti, Q. Wang, C.D.J. Tavares [et al.] //Bioorg. Med. Chem. – 2014. – Vol. 22. – P. 4910-4916.298. Synthesis and discovery of N-carbonylpyrrolidine- or N-sulfonylpyrrolidinecontaining uracil derivatives as potent human deoxyuridine triphosphatase inhibitors / H. Miyakoshi, S. Miyahara, T.
Yokogawa [et al.] // J. Med. Chem. – 2012. –Vol. 55. – P. 2960-2969.299. Synthesis and evaluation as PDE4 inhibitors of pyrimidine-2,4-dione deriva-383tives / M.P. Goivannoni, A. Graziano, R. Matucci [et al.] // Drud Dev. Res. –2011. – Vol. 72. – P. 274-288.300. Synthesis and evaluation of double-prodrugs against HIV. Conjugation of D4Twith 6-benzyl-1-(ethoxymethyl)-5-isopropyluracil (MKC-442, Emivirine)-typereverse transcriptase inhibitors via the SATE approach / L.
Petersen, P. T. Jorgensen, C. Nielsen [et al.] // J. Med. Chem. – 2005. – Vol. 35. – P. 1211-1220.301. Synthesis and evaluation of new potential HIV-1 non-nucleoside reverse transcriptase inhibitors. New analogues of MKC-442 containing Michael acceptors inthe C-6 position / L. Petersen, C.
H. Jessen, E. B. Pedersen, C. Nielsen // Org. Biomol. Chem. – 2003. – № 1. – P. 3541-3545.302. Synthesis and evaluation of novel 3-(3,5-dimethylbenzyl)uracil analogs as potential anti-HIV-1 agents / N. Sakakibara, T. Hamasaki, M. Baba [et al.] // Bioorg.Med.
Chem. – 2013 – Vol. 21. – P. 5900-5906.303. Synthesis and evaluation of organosilicon inhibitors of active purine transportin human osteoblasts / S. Ciro, C. Rubio, K. Estieu-Gionnet [et al.] // ChemBioChem. – 2002. - № 3. – P. 341-347.304. Synthesis and in vitro antiproliferative evaluation of novel N-alkylated 6isobutil- and propyl pyrimidine derivatives / T. Gazivoda Kraljevic, N. Ilic, V.Stepanic [et al.] // Bioorg. Med. Chem.
Lett. – 2014. – Vol. 24. – P. 2913-2917.305. Synthesis and pharmacology activity willadiine derivativesacting as antagonistof kainate receptors / N.P. Dolman, H.M. Troop, J.C. More [et al.] // J. Med.Chem. – 2005. – Vol. 48. – P. 7867-7881.306. Synthesis and pharmacological characterization of N3-substituted willardiinederivatives: role of the substituent at the 5-position of the uracil ring in the development of highly potent and selective GLUK5 kainate receptor antagonists / N.P.Dolman, J.C.A. More, A. Alt [et al.] // J. Med. Chem.
– 2007. – Vol. 50. – P.1558-1570.307. Synthesis and SAR oh highly potent and selective dopamine D3-receptor antagonists: 1H-pyrimidine-2-one derivatives / H. Geneste, G. Backfisch, W. Braje[et al.] // Bioorg. Med. Chem. Lett. – 2006. – Vol. 16. – P. 490-494.384308. Synthesis and structrural studies of three uracil derivatives, methyl 3-(2,4dioxo-3,4-dihydropyrimidin-1(2H)-yl)propanate, methyl 3-(5-nitro-2,4-dioxo-3,4dihydropyrimidin-1(2H)-yl)propanateandethyl3-(5-nitro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)propanate / W.
Liu, X. Feng, Y. Tao [et al.] // J.Chem. Crystallogrm. – 2014. – Vol. 44. – P. 597-603.309. Synthesis, cytostatic and anti-HIV evaluations of the new unsaturated acyclicC-5 pyrimidine nucleoside analogues / T. Gazivoda, S. Raic-Malic, V. Kristafor[et al.] // Bioorg. Med. Chem. – 2008. – Vol. 16. – P. 5624-5634.310. Synthetic electroorganic chemistry. 14. Synthesis of 5-fluorouracil derivativeshaving N-acylazacycloalkanes and lactams / T. Nishitani, H. Horikawa, T.
Iwasaki [et al.] // J. Org. Chem. – 1982. - Vol. 47. - Р. 1706-1712.311. Synthesis, evaluation and molecular docking of prolyl-fluoropyrrolidine derivatives as dipeptidyl peptidase IV inhibitors / М. Sharma, M. Gupta, D. Singh [etal.] // Chem. Biol. Drug Des. - 2013. - Vol. 82. - P. 156-166.312. Synthesis of 1-(alkoxymethyl)-5-benzyl-6-methyluracil as potential nonnucleoside HIV-1 RT inhibitors / Y. Chen, Y. Guo, H. Yang [et al.] // Synth.
Commun. –2006. – Vol. 36. – P. 2913-2920.313. Synthesis of 6-alkyluridines from 6-cyanouridine via Zinc(II) chloridecatalyzed nucleophilic substitution with alkyl Grignard reagents / Yu-Ch. Shih,Ya-Y. Yang, C.-C. Lin, Y.-C. Chein // J. Org. Chem. – 2013. – Vol. 78. – P.4027-4036.314. Synthesis of 1-arylated derivatives of 5-fluorouracil as potential antitumordrugs / J. You, Sh. Chen, Y, Wang, Y.
